Short descriptionPotent, selective PKC inhibitor
Biological descriptionPotent and selective protein kinase C (PKC) inhibitor (IC = 15 nM). Displays selectivity for PKC-α and PKC-β1 over PKC-βII, PKC-γ and PKC-ε (IC50 values are 8, 8, 14, 13, and 39 nM respectively). Also potent CDK2 antagonist (IC50 = 200 nM).
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ImportantThis product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.