Write Your Own Review
You're reviewing:I-CBP 112
Rate this item:

Biological Data

Biological description CBP/p300 Bromodomain inhibitor (IC50 values are 170 and 625 nM). Selective over ATAD2, BAZ2B, BRD2, BRD4, PB1, PCAF, PHIP and TRIM24/TIF-1a. Shows accelerated FRAP recovery at 1 µM.

Solubility & Handling

Storage instructions +4°C
Solubility overview Soluble in DMSO (100mM)
Important This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.

Calculators

Molarity

=
x
x
More Info

Dilution

x
=
x
More Info

Chemical Data

Purity >98%
Chemical name 1-[7-(3,4-Dimethoxyphenyl)-9-[[(3S)-1-methylpiperidin-3-yl]methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
Molecular Weight 468.59
Chemical structure I-CBP 112 Chemical Structure
Molecular Formula C27H36N2O5
CAS Number 1640282-31-0
PubChem identifier 90488984
SMILES COC(C(OC)=C1)=CC=C1C2=CC(OC[C@H]3CCCN(C)C3)=C(OCCN(C(CC)=O)C4)C4=C2
InChiKey YKNAKDFZAWQEEO-IBGZPJMESA-N

References for I-CBP 112

References are publications that support the biological activity of the product

1 Item