Product overview

  • Name
    LE 300
  • Short description
    Potent, selective D1 receptor antagonist
  • Biological description
    Potent and selective D1 receptor antagonist (Ki values are 0.08 - 1.9 nM and 6 - 45 nM for D1 and D2 receptors respectively). Also shows activity at the 5-HT2A receptor (Ki = 20 nM). Active in vivo.
  • Biological action
    Antagonist
  • Purity
    >98%
  • Our products in action

Properties

  • Chemical name
    6,7,8,9,14,15-Hexahydro-7-methyl-5H -indolo[3,2-f][3]benzazecine
  • Molecular Weight
    290.41
  • Molecular Formula
    C20H22N2
  • CAS Number
    274694-98-3

Storing and Using Your Product

  • Storage instructions
    room temperature
  • Solubility overview
    soluble in DMSO (100mM) or water (50mM, 1eq. HCl)
  • Important
    This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.

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