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Tertiapin LQ

(HB1107)
Data

Product overview

  • Name
    Tertiapin LQ
  • Short description
    Potent, selective Kir1.1 channel blocker
  • Biological description
    Tertiapin-Q derivative. Potent and selective Kir1.1 channel blocker. Selective for Kir1.1 over Kir3.1/3.2 and Kir3.1/3.4 (Kd values are 1.1, 274 and 361 nM respectively).
  • Biological action
    Blocker
  • Citations

Properties

  • Molecular Weight
    2428.03
  • Molecular Formula
    C106H179N33O24S4
  • PubChem identifier
    90488935
  • SMILES
    [H]N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H]1CSSC[C@@H]2NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]3CCCN3C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC3=CNC4=C3C=CC=C4)NC2=O)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@H](CC(N)=O)NC1=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC
  • InChiKey
    WUMIWMIQOSXVPZ-ZPWFPUPGSA-N

Storing and Using Your Product

  • Storage instructions
    -20°C
  • Solubility overview
    soluble in acetonitrile (2mg/ml)
  • Important
    This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.

References for Tertiapin LQ

  • Engineered specific and high-affinity inhibitor for a subtype of inward-rectifier K+ channels.

    Ramu Y et al (2008) Proc Natl Acad Sci U S A 105(31) : 10774-8.
    PubMedID: 18669667
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