WAY 100635 maleate
(HB1790)
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Code: HB1643
Pack: 10mg,50mg
Code: HB1812
Pack: 10mg,50mg
Code: HB1858
Pack: 10mg,25mg
WAY 100635 maleate
(HB1790)- Data
- Support & Resources
Product overview
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Name
WAY 100635 maleate
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Short description
Potent 5-HT1A receptor antagonist. D4 receptor agonist.
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Biological description
Potent 5-HT1A receptor antagonist (IC50 value = 2.2 nM). More than 100-fold selective for 5-HT1A compared with other 5-HT receptors. Also acts as an agonist at D4 receptor (IC50 value = 16 nM). Active in vivo.
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Biological action
Antagonist
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Purity
>99%
- Citations
Properties
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Chemical name
N-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinylcyclohexanecarboxamide maleate
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Molecular Weight
538.64
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Chemical structure
![WAY 100635 maleate [634908-75-1]](data:image/gif;base64,R0lGODlhAQABAAD/ACwAAAAAAQABAAACADs= "WAY 100635 maleate [634908-75-1]")
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Molecular Formula
C25H34N4O2.C4H4O4
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CAS Number
634908-75-1
![WAY 100635 maleate [634908-75-1]](https://www.hellobio.com/media/catalog/product/cache/1/image/9df78eab33525d08d6e5fb8d27136e95/h/b/hb1790.png "WAY 100635 maleate [634908-75-1]")
Storing and Using Your Product
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Storage instructions
room temperature (desiccate)
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Important
This product is for RESEARCH USE ONLY and is not intended for therapeutic or diagnostic use. Not for human or veterinary use.
References for WAY 100635 maleate
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A pharmacological profile of the selective silent 5-HT1A receptor antagonist, WAY-100635.
Forster EA et al (1995) Eur J Pharmacol 281(1) : 81-8.PubMedID: 8566121 -
WAY-100635 is a potent dopamine D4 receptor agonist.
Chemel BR et al (2006) Psychopharmacology (Berl) 188(2) : 244-51.PubMedID: 16915381 -
WAY 100635 produces discriminative stimulus effects in rats mediated by dopamine D(4) receptor activation.
Marona-Lewicka D et al (2009) Behav Pharmacol 20(1) : 114-8.PubMedID: 19179855
Reviews & Product Guides
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