Agonists & activators

An agonist or activator, is a drug or chemical that binds to and activates a protein, such as receptor or enzyme. Full agonists have high efficacy, eliciting a full response whilst occupying a small proportion of receptors. Partial agonists have a lower efficacy and cannot produce a maximal response, even if occupying a high proportion of receptors. Inverse agonists can bind to the same receptor binding-site as an agonist, but elicit an opposite effect. Researchers can save up to 50% on activators, agonists, partial agonists and inverse agonists from Hello Bio - they are up to half the price of other suppliers.

  1. Description:

    Synthetic prostaglandin E2 derivative. Induces stem cell proliferation.

    Purity :

    >98%

    16,16-Dimethyl Prostaglandin E2
    Pack: Price: Qty:
    1mg
    $93
  2. Description:

    5-HT4 receptor agonist and 5-HT3 antagonist

    Pack: Price: Qty:
    5mg
    $57
  3. A 769662(HB1351)

    Description:

    Potent, reversible AMPK activator. Inhibits MSC proliferation.

    Purity :

    >98%

    A 769662
    Pack: Price: Qty:
    10mg
    $136
    50mg
    $528
  4. Description:

    Potent dopamine D4 receptor partial agonist

    Purity :

    >99%

    Pack: Price: Qty:
    50mg
    $451
  5. Description:

    GABA receptor agonist and glutamergic modulator

    Acamprosate calcium
    Pack: Price: Qty:
    100mg
    $160
  6. ACBC(HB0100)

    Description:

    Competitive NMDA receptor partial agonist

    ACBC
    Pack: Price: Qty:
    1g
    $90
    5g
    $330
  7. AdipoRon(HB3738)

    Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $267
  8. Description:

    AdipoR1 and AdipoR2 agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $312
  9. Aftin-4(HB3741)

    Description:

    Roscovitine-related purine with no activity on CDKs. Roscovitine control. Increases Aβ42 production.

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $171
  10. Aftin-5(HB3742)

    Description:

    Roscovitine-related purine with no activity on CDKs. Roscovitine control. Increases Aβ42 production.

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $209
  11. AICAR(HB2152)

    Description:

    AMPK activator. Promotes osteogenic differentiation of bone marrow-derived MSCs.

    Purity :

    >99%

    AICAR
    Pack: Price: Qty:
    25mg
    $55
  12. Description:

    Potent GABAA receptor positive allosteric modulator

    Allopregnanolone
    Pack: Price: Qty:
    50mg
    $558
  13. Description:

    Immunostimulant. Natural killer T cell stimulator.

    Purity :

    >96%

    Pack: Price: Qty:
    1mg
    $261
  14. (S)-AMPA(HB0052)

    Description:

    AMPA receptor agonist

    Purity :

    >99%

    AMPAR mediated whole cell current in response to S-AMPA
    Pack: Price: Qty:
    1mg
    $71
    5mg
    $186
  15. (R,S)-AMPA(HB0030)

    Description:

    Prototypic AMPA receptor agonist

    Purity :

    >98%

    (R,S)-AMPA
    Pack: Price: Qty:
    10mg
    $104
    50mg
    $421
  16. Description:

    Potent nicotinic agonist

    Purity :

    >96%

    Pack: Price: Qty:
    1mg
    $136
  17. Aniracetam(HB0116)

    Description:

    Nootrophic AMPA receptor positive allosteric modulator

    Purity :

    >99%

    Aniracetam
    Pack: Price: Qty:
    100mg
    $218
    500mg
    $870
  18. L-AP4(HB0370)

    Description:

    Selective group III mGluR agonist. Inhibits synaptic transmission.

    Purity :

    >99%

    L-AP4
    Pack: Price: Qty:
    5mg
    $56
    10mg
    $102
    25mg
    $227
    50mg
    $415
  19. Description:

    Caspase activator

    Purity :

    >99%

    Pack: Price: Qty:
    50mg
    $441
  20. Description:

    NMDA receptor agonist

    D-Aspartic acid
    Pack: Price: Qty:
    1g
    $75
  21. (S)-ATPA(HB0854)

    Description:

    Selective GluK1 kainate / AMPA receptor agonist

    Pack: Price: Qty:
    5mg
    $160
  22. (R)-Baclofen(HB0952)

    Description:

    Selective GABAB receptor agonist

    Purity :

    >99%

    Reversible inhibition of EPSC amplitude and increased EPSC paired pulse ration in response to Baclofen
    Pack: Price: Qty:
    10mg
    $44
    50mg
    $184
  23. Description:

    Selective GABAB receptor agonist

    Purity :

    >99%

    (RS)-Baclofen
    Pack: Price: Qty:
    1g
    $59
  24. Description:

    L-type Ca2+ channel agonist. Aids iPSCs generation from Mouse embryonic fibroblasts.

    Purity :

    >99%

    (±)-Bay K 8644
    Pack: Price: Qty:
    10mg
    $129
    50mg
    $506
  25. BINA(HB0133)

    Reviews:
    Description:

    Potent, selective mGlu2 positive allosteric modulator

    Purity :

    >98%

    BINA
    Pack: Price: Qty:
    5mg
    $96
    10mg
    $142
    25mg
    $283
  26. Description:

    5-HT1A partial agonist

    Pack: Price: Qty:
    10mg
    $59
    50mg
    $216
  27. Bradykinin(HB3101)

    Description:

    Endogenous bradykinin receptors agonist

    Purity :

    >95%

    Pack: Price: Qty:
    5mg
    $23
    25mg
    $91
  28. BRL 54443(HB1664)

    Description:

    Potent 5-ht1E/1F receptor agonist

    Pack: Price: Qty:
    10mg
    $103
    50mg
    $354
  29. Description:

    Classic 5-HT1A partial agonist

    Purity :

    >99%

    Pack: Price: Qty:
    100mg
    $54
  30. Description:

    Ceramide-activated protein phosphatase (CAPP) activator

    Pack: Price: Qty:
    5mg
    $268
  31. Description:

    Nonpsychoactive cannabinoid found in cannabis

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $80
    50mg
    $300
  32. Description:

    TRPV1 channel agonist

    Purity :

    >98%

    (E)-Capsaicin
    Pack: Price: Qty:
    50mg
    $51
    250mg
    $203
  33. CDPPB(HB0175)

    Description:

    Selective mGlu5 positive allosteric modulator

    Purity :

    >98%

    CDPPB
    Pack: Price: Qty:
    10mg
    $122
    50mg
    $490
  34. Description:

    Potent STING ligand

    Purity :

    >98%

    Pack: Price: Qty:
    500μg
    $219
  35. Description:

    Selective mGluR5 agonist. Water soluble sodium salt.

    Purity :

    >99%

    (R,S)-CHPG sodium salt
    Pack: Price: Qty:
    10mg
    $65
    50mg
    $269
  36. (R,S)-CHPG(HB0033)

    Description:

    Selective mGlu5 agonist

    Purity :

    >98%

    (R,S)-CHPG
    Pack: Price: Qty:
    10mg
    $59
    50mg
    $252
  37. Ciglitazone(HB2551)

    Description:

    Selective PPARγ agonist

    Purity :

    >99%

    Pack: Price: Qty:
    25mg
    $331
  38. Description:

    Selective mGlu4 agonist

    Purity :

    >98%

    Cinnabarinic acid
    Pack: Price: Qty:
    10mg
    $167
    50mg
    $668
    100mg
    $1,003
  39. CIQ(HB0197)

    Reviews:
    Description:

    GluN2C / GluN2D subunit selective NMDA receptor positive allosteric modulator

    Purity :

    >98%

    CIQ
    Pack: Price: Qty:
    10mg
    $122
  40. Citrinin(HB3839)

    Description:

    Mitochondrial permeability transition pore (MPTP) activator

    Purity :

    >97%

    Pack: Price: Qty:
    25mg
    $267
  41. Clozapine(HB1607)

    Description:

    Prototypic, atypical antipsychotic, binds to both serotonin and dopamine receptors

    Purity :

    >99%

    Clozapine
    Pack: Price: Qty:
    50mg
    $85
    500mg
    $350
  42. Reviews:
    Description:

    Water soluble prototypical DREADD activator. Clozapine metabolite.

    Purity :

    >98%

    Clozapine N-oxide (CNO) (water soluble)
    Pack: Price: Qty:
    5mg
    $50
    10mg
    $85
    25mg
    $185
    100mg
    $650
  43. Description:

    Highly potent hM3Dq DREADD agonist

    Purity :

    >98%

    Compound 21 (DREADD agonist 21)
    Pack: Price: Qty:
    5mg
    $55
    10mg
    $98
    25mg
    $225
    100mg
    $820
  44. Description:

    Highly potent hM3Dq DREADD agonist. Water soluble.

    Purity :

    >98%

    Compound 21 (DREADD agonist 21) hydrochloride (water soluble)
    Pack: Price: Qty:
    5mg
    $63
    10mg
    $113
    25mg
    $259
    100mg
    $943
  45. Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $323
  46. Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $323
  47. Description:

    Endogenous gluococorticoid. MR and GR agonist.

    Purity :

    >99%

    Corticosterone
    Pack: Price: Qty:
    100mg
    $74
  48. Description:

    Potent, selective 5-HT1B receptor agonist

    Purity :

    >98%

    CP 94253 hydrochloride
    Pack: Price: Qty:
    10mg
    $136
    50mg
    $499
  49. Description:

    AMPA receptor positive allosteric modulator. Inhibits AMPAR desensitization.

    Purity :

    >98%

    Cyclothiazide inhibition of AMPA receptor mediated EPSCs
    Pack: Price: Qty:
    10mg
    $43
    50mg
    $184
  50. CyPPA(HB1044)

    Description:

    Selective KCa2.2 / KCa2.3 activator

    Purity :

    >99%

    CyPPA
    Pack: Price: Qty:
    10mg
    $125
    50mg
    $502