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Agonists & activators

An agonist or activator, is a drug or chemical that binds to and activates a protein, such as receptor or enzyme. Full agonists have high efficacy, eliciting a full response whilst occupying a small proportion of receptors. Partial agonists have a lower efficacy and cannot produce a maximal response, even if occupying a high proportion of receptors. Inverse agonists can bind to the same receptor binding-site as an agonist, but elicit an opposite effect. Researchers can save up to 50% on activators, agonists, partial agonists and inverse agonists from Hello Bio - they are up to half the price of other suppliers.

  1. 16,16-Dimethyl Prostaglandin E2
    Description:

    Synthetic prostaglandin E2 derivative. Induces stem cell proliferation.

    Purity :

    >98%

  2. Description:

    5-HT4 receptor agonist and 5-HT3 antagonist

  3. A 769662

    A 769662(HB1351)

    Description:

    Potent, reversible AMPK activator. Inhibits MSC proliferation.

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $136
    50mg
    $528
  4. Description:

    Potent dopamine D4 receptor partial agonist

    Purity :

    >99%

    Pack: Price: Qty:
    50mg
    $451
  5. Acamprosate calcium
    Description:

    GABA receptor agonist and glutamergic modulator

    Pack: Price: Qty:
    100mg
    $160
  6. ACBC

    ACBC(HB0100)

    Description:

    Competitive NMDA receptor partial agonist

    Pack: Price: Qty:
    1g
    $90
    5g
    $330
  7. AdipoRon(HB3738)

    Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $267
  8. Description:

    AdipoR1 and AdipoR2 agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $312
  9. Aftin-4(HB3741)

    Description:

    Roscovitine-related purine with no activity on CDKs. Roscovitine control. Increases Aβ42 production.

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $171
  10. Aftin-5(HB3742)

    Description:

    Roscovitine-related purine with no activity on CDKs. Roscovitine control. Increases Aβ42 production.

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $209
  11. AICAR

    AICAR(HB2152)

    Description:

    AMPK activator. Promotes osteogenic differentiation of bone marrow-derived MSCs.

    Purity :

    >99%

    Pack: Price: Qty:
    25mg
    $55
  12. Allopregnanolone
    Description:

    Potent GABAA receptor positive allosteric modulator

    Pack: Price: Qty:
    50mg
    $558
  13. Description:

    Immunostimulant. Natural killer T cell stimulator.

    Purity :

    >96%

    Pack: Price: Qty:
    1mg
    $261
  14. AMPAR mediated whole cell current in response to S-AMPA

    (S)-AMPA(HB0052)

    Description:

    AMPA receptor agonist

    Purity :

    >99%

    Pack: Price: Qty:
    1mg
    $71
    5mg
    $186
  15. (R,S)-AMPA

    (R,S)-AMPA(HB0030)

    Description:

    Prototypic AMPA receptor agonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $104
    50mg
    $421
  16. Description:

    Potent nicotinic agonist

    Purity :

    >96%

    Pack: Price: Qty:
    1mg
    $136
  17. Aniracetam

    Aniracetam(HB0116)

    Description:

    Nootrophic AMPA receptor positive allosteric modulator

    Purity :

    >99%

    Pack: Price: Qty:
    100mg
    $218
    500mg
    $870
  18. L-AP4

    L-AP4(HB0370)

    Reviews:
    Description:

    L-AP4 is a selective group III mGluR agonist which inhibits synaptic transmission.

    Purity :

    >99%

    Pack: Price: Qty:
    5mg
    $56
    10mg
    $102
    25mg
    $227
    50mg
    $415
  19. Description:

    Caspase activator

    Purity :

    >99%

    Pack: Price: Qty:
    50mg
    $441
  20. D-Aspartic acid
    Description:

    NMDA receptor agonist

  21. (S)-ATPA(HB0854)

    Description:

    Selective GluK1 kainate / AMPA receptor agonist

    Pack: Price: Qty:
    5mg
    $160
  22. Reversible inhibition of EPSC amplitude and increased EPSC paired pulse ration in response to Baclofen

    (R)-Baclofen(HB0952)

    Description:

    Selective GABAB receptor agonist

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $44
    50mg
    $184
  23. (RS)-Baclofen

    (RS)-Baclofen(HB0953)

    Description:

    Selective GABAB receptor agonist

    Purity :

    >99%

  24. (±)-Bay K 8644
    Description:

    L-type Ca2+ channel agonist. Aids iPSCs generation from Mouse embryonic fibroblasts.

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $129
    50mg
    $506
  25. BINA

    BINA(HB0133)

    Reviews:
    Description:

    Potent, selective mGlu2 positive allosteric modulator

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $96
    10mg
    $142
    25mg
    $283
  26. Description:

    5-HT1A partial agonist

    Pack: Price: Qty:
    10mg
    $59
    50mg
    $216
  27. Bradykinin(HB3101)

    Description:

    Endogenous bradykinin receptors agonist

    Purity :

    >95%

    Pack: Price: Qty:
    5mg
    $23
    25mg
    $91
  28. BRL 54443(HB1664)

    Description:

    Potent 5-ht1E/1F receptor agonist

    Pack: Price: Qty:
    10mg
    $103
    50mg
    $354
  29. Description:

    Classic 5-HT1A partial agonist

    Purity :

    >99%

    Pack: Price: Qty:
    100mg
    $54
  30. Description:

    Ceramide-activated protein phosphatase (CAPP) activator

    Pack: Price: Qty:
    5mg
    $268
  31. Description:

    Nonpsychoactive cannabinoid found in cannabis

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $80
    50mg
    $300
  32. (E)-Capsaicin

    (E)-Capsaicin(HB1179)

    Description:

    TRPV1 channel agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $51
    250mg
    $203
  33. CDPPB

    CDPPB(HB0175)

    Description:

    Selective mGlu5 positive allosteric modulator

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $122
    50mg
    $490
  34. Description:

    Potent STING ligand

    Purity :

    >98%

    Pack: Price: Qty:
    500μg
    $219
  35. (R,S)-CHPG sodium salt
    Description:

    Selective mGluR5 agonist. Water soluble sodium salt.

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $65
    50mg
    $269
  36. (R,S)-CHPG

    (R,S)-CHPG(HB0033)

    Description:

    Selective mGlu5 agonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $59
    50mg
    $252
  37. Ciglitazone(HB2551)

    Description:

    Selective PPARγ agonist

    Purity :

    >99%

    Pack: Price: Qty:
    25mg
    $331
  38. Cinnabarinic acid
    Description:

    Selective mGlu4 agonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $167
    50mg
    $668
    100mg
    $1,003
  39. CIQ

    CIQ(HB0197)

    Reviews:
    Description:

    GluN2C / GluN2D subunit selective NMDA receptor positive allosteric modulator

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $122
  40. Citrinin(HB3839)

    Description:

    Mitochondrial permeability transition pore (MPTP) activator

    Purity :

    >97%

    Pack: Price: Qty:
    25mg
    $267
  41. Clozapine

    Clozapine(HB1607)

    Description:

    Prototypic, atypical antipsychotic, binds to both serotonin and dopamine receptors

    Purity :

    >99%

    Pack: Price: Qty:
    50mg
    $85
    500mg
    $350
  42. Clozapine dihydrochloride (water soluble)
    Reviews:
    Description:

    Water soluble prototypic, atypical antipsychotic. Binds to both serotonin and dopamine receptors.

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $37
    50mg
    $96
  43. Clozapine N-oxide (CNO) (freebase)
    Reviews:
    Description:

    Prototypical DREADD activator. Clozapine metabolite.

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $50
    10mg
    $85
    25mg
    $185
    100mg
    $650
  44. Clozapine N-oxide (CNO) dihydrochloride (water soluble)
    Reviews:
    Description:

    Dihydrochloride salt of CNO - the prototypical DREADD activator

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $45
    10mg
    $77
    25mg
    $167
    100mg
    $585
  45. Compound 21 (DREADD agonist 21)
    Description:

    Highly potent hM3Dq DREADD agonist

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $55
    10mg
    $98
    25mg
    $225
    100mg
    $820
  46. Compound 21 (DREADD agonist 21) hydrochloride (water soluble)
    Description:

    Highly potent hM3Dq DREADD agonist. Water soluble.

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $63
    10mg
    $113
    25mg
    $259
    100mg
    $943
  47. Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $323
  48. Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $323
  49. Corticosterone
    Description:

    Endogenous gluococorticoid. MR and GR agonist.

    Purity :

    >99%

    Pack: Price: Qty:
    100mg
    $74
  50. CP 94253 hydrochloride
    Description:

    Potent, selective 5-HT1B receptor agonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $136
    50mg
    $499