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G protein coupled receptors

G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. GPCRs include acetycholine muscarinic, adenosine, GABAB, and histamine receptors, and the metabotropic glutamate receptors (Group I, Group II and Group III). Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

  1. Description:

    5-HT4 receptor agonist and 5-HT3 antagonist

    Pack: Price: Qty:
    5mg
    $57
  2. 6-Hydroxydopamine (6-OHDA) hydrobromide
    Description:

    Neurotoxin, widely used to produce the 6-OHDA Parkinson’s disease model

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $27
    250mg
    $80
    1g
    $265
  3. Description:

    Potent dopamine D4 receptor partial agonist

    Purity :

    >99%

    Pack: Price: Qty:
    50mg
    $451
  4. Acamprosate calcium
    Description:

    GABA receptor agonist and glutamergic modulator

    Pack: Price: Qty:
    100mg
    $160
  5. Description:

    Serotonin N-acetyltransferase substrate

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $91
    50mg
    $332
  6. Adenosine

    Adenosine(HB2843)

    Description:

    Endogenous adenosine receptor agonist

    Pack: Price: Qty:
    50mg
    $49
  7. AdipoRon(HB3738)

    Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $267
  8. Description:

    AdipoR1 and AdipoR2 agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $312
  9. AF-DX 116

    AF-DX 116(HB1501)

    Description:

    Selective, competitive M2 receptor antagonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $185
    50mg
    $700
  10. Description:

    Non-selective β-adrenoceptor antagonist. Also a 5-HT1A receptor antagonist.

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $71
  11. AM251(HB2776)

    Reviews:
    Description:

    Potent, selective CB1 receptor antagonist / inverse agonist

    Purity :

    >98%

    Pack: Price: Qty:
    1mg
    $41
    10mg
    $87
    50mg
    $366
  12. AM 281

    AM 281(HB2312)

    Description:

    Potent, selective CB1 receptor antagonist / inverse agonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $115
    50mg
    $475
  13. Amauromine(HB3758)

    Description:

    Potent and selective CB1 receptor antagonist

    Purity :

    >95%

    Pack: Price: Qty:
    1mg
    $144
  14. AMD 3100 octahydrochloride
    Description:

    Potent, selective CXCR4 antagonist. Mobilizes hematopoietic stem cells.

    Pack: Price: Qty:
    10mg
    $107
  15. Amisulpride(HB1879)

    Description:

    Potent, selective dopamine D2 and D3 receptor antagonist. Atypical antipsychotic.

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $93
  16. L-AP4

    L-AP4(HB0370)

    Reviews:
    Description:

    L-AP4 is a selective group III mGluR agonist which inhibits synaptic transmission.

    Purity :

    >99%

    Pack: Price: Qty:
    5mg
    $56
    10mg
    $102
    25mg
    $227
    50mg
    $415
  17. Reversible inhibition of EPSC amplitude and increased EPSC paired pulse ration in response to Baclofen

    (R)-Baclofen(HB0952)

    Description:

    Selective GABAB receptor agonist

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $44
    50mg
    $184
  18. (RS)-Baclofen

    (RS)-Baclofen(HB0953)

    Description:

    Selective GABAB receptor agonist

    Purity :

    >99%

  19. BINA

    BINA(HB0133)

    Reviews:
    Description:

    Potent, selective mGlu2 positive allosteric modulator

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $96
    10mg
    $142
    25mg
    $283
  20. Description:

    5-HT1A partial agonist

    Pack: Price: Qty:
    10mg
    $59
    50mg
    $216
  21. Description:

    Potent, selective endothelin receptor A (ETA) antagonist

    Purity :

    >98%

    Pack: Price: Qty:
    5mg
    $361
  22. Description:

    Potent, selective endothelin B receptor (ETBR) antagonist

    Purity :

    >95%

    Pack: Price: Qty:
    500μg
    $152
    1mg
    $200
  23. Bradykinin(HB3101)

    Description:

    Endogenous bradykinin receptors agonist

    Purity :

    >95%

    Pack: Price: Qty:
    5mg
    $23
    25mg
    $91
  24. Description:

    Selective h5-HT1D antagonist

    Pack: Price: Qty:
    10mg
    $119
    50mg
    $451
  25. BRL 54443(HB1664)

    Description:

    Potent 5-ht1E/1F receptor agonist

    Pack: Price: Qty:
    10mg
    $103
    50mg
    $354
  26. Description:

    Classic 5-HT1A partial agonist

    Purity :

    >99%

    Pack: Price: Qty:
    100mg
    $54
  27. CA200623 CellAura fluorescent adenosine agonist [NECA]
    Description:

    Fluorescent adenosine receptor agonist

    Pack: Price: Qty:
    50μg
    $189
  28. CA200634 CellAura fluorescent adenosine antagonist [XAC]
    Description:

    Competitive fluorescent adenosine receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  29. CA200645 CellAura fluorescent adenosine A3 antagonist [XAC]
    Description:

    Fluorescent A3 adenosine receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  30. CA200656 CellAura fluorescent β2 antagonist [(±)-propranolol]
    Description:

    Fluorescent β2 adrenoceptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  31. CA200689 CellAura fluorescent β2 antagonist [(S)-propranolol-red]
    Description:

    Competitive fluorescent β2-adrenoceptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  32. CA200693 CellAura fluorescent β2 antagonist [(S)-propranolol-green]
    Description:

    Fluorescent β2-adrenoceptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  33. CA200773 CellAura fluorescent D1 antagonist [SKF83566-green]
    Description:

    Fluorescent D1 dopamine receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  34. CA200799 CellAura fluorescent H1 antagonist [mepyramine]
    Description:

    Fluorescent H1 histamine receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  35. CA200821 CellAura fluorescent H2 antagonist [aminopotentidine]
    Description:

    Fluorescent H2 histamine receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  36. CA200843 CellAura fluorescent H3 antagonist [clobenpropit]
    Description:

    Fluorescent H3 histamine receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  37. Description:

    Fluorescent GABAB receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  38. CA200992 CellAura fluorescent 5-HT1A antagonist [NAN-190]
    Description:

    Fluorescent 5-HT1A receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  39. Description:

    Fluorescent 5-HT2A receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  40. Description:

    Fluorescent muscarinic M1 receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  41. Description:

    Fluorescent D3 antagonist [piperidinyl pyrazole-red]

    Pack: Price:
    50μg
    $189
    -
  42. Description:

    Fluorescent muscarinic M2 antagonist [benzylidine-red-2]

    Pack: Price: Qty:
    50μg
    $189
  43. Description:

    Fluorescent D3 antagonist [BP897-red]

    Pack: Price:
    50μg
    $189
    -
  44. Description:

    Fluorescent muscarinic M4 receptor antagonist

    Pack: Price: Qty:
    50μg
    $189
  45. Caffeine

    Caffeine(HB2846)

    Description:

    Non-selective, competitive adenosine receptor antagonist / PDE inhibitor

    Pack: Price: Qty:
    100mg
    $42
  46. (-)-Cannabidiol(HB2785)

    Description:

    Nonpsychoactive cannabinoid found in cannabis

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $80
    50mg
    $300
  47. CDPPB

    CDPPB(HB0175)

    Description:

    Selective mGlu5 positive allosteric modulator

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $93
    50mg
    $388
  48. CGP 35348

    CGP 35348(HB0955)

    Description:

    Selective GABAB receptor antagonist

    Pack: Price: Qty:
    10mg
    $138
  49. CGP55845 hydrochloride
    Reviews:
    Description:

    Potent, selective GABAB receptor antagonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $113
    50mg
    $465
  50. 2-Chloroadenosine (CADO)
    Description:

    Adenosine receptor agonist

    Purity :

    >99%

    Pack: Price: Qty:
    250mg
    $283
    1g
    $725