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G protein coupled receptors

G-protein-coupled receptors (also known as GPCRs, transmembrane receptors, or 7-TM receptors), are integral membrane proteins that contain seven membrane-spanning domains (helices). They are coupled to heterotrimeric G proteins on the intracellular side of the cell membrane. Ligand binding causes a conformational change in the GPCR, that is then transmitted to the G protein, activating a signal transduction pathway. GPCRs include acetycholine muscarinic, adenosine, GABAB, and histamine receptors, and the metabotropic glutamate receptors (Group I, Group II and Group III). Researchers can save up to 50% on GPCR receptor agonists, antagonists and allosteric modulators from Hello Bio - they are up to half the price of other suppliers.

  1. Description:

    5-HT4 receptor agonist and 5-HT3 antagonist

    Pack: Price: Qty:
    5mg
    $57
  2. 6-Hydroxydopamine (6-OHDA) hydrobromide
    Description:

    Neurotoxin, widely used to produce the 6-OHDA Parkinson’s disease model

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $27
    250mg
    $80
    1g
    $265
  3. Description:

    Potent dopamine D4 receptor partial agonist

    Purity :

    >99%

    Pack: Price: Qty:
    50mg
    $451
  4. Acamprosate calcium
    Description:

    GABA receptor agonist and glutamatergic modulator

    Pack: Price: Qty:
    100mg
    $160
  5. Description:

    Serotonin N-acetyltransferase substrate

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $91
    50mg
    $332
  6. Adenosine

    Adenosine(HB2843)

    Description:

    Endogenous adenosine receptor agonist

    Pack: Price: Qty:
    50mg
    $49
  7. AdipoRon(HB3738)

    Description:

    Adiponectin receptor (AdipoR) agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $267
  8. Description:

    AdipoR1 and AdipoR2 agonist

    Purity :

    >98%

    Pack: Price: Qty:
    50mg
    $312
  9. AF-DX 116

    AF-DX 116(HB1501)

    Description:

    Selective, competitive M2 receptor antagonist

    Purity :

    >98%

    Pack: Price: Qty:
    10mg
    $185
    50mg
    $700
  10. Description:

    Non-selective β-adrenoceptor antagonist. Also a 5-HT1A receptor antagonist.

    Purity :

    >99%

    Pack: Price: Qty:
    10mg
    $71